Laufer, Radoslaw

The discovery of PLK4 inhibitors: (E)-3-((1H-Indazol-6-yl)methylene)indolin-2-ones as novel antiproliferative agents. [electronic resource] - Journal of medicinal chemistry Aug 2013 - 6069-87 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1520-4804

10.1021/jm400380m doi


Animals
Antineoplastic Agents--chemical synthesis
Cell Cycle--drug effects
Cell Line, Tumor
Cell Proliferation--drug effects
Drug Screening Assays, Antitumor
Female
Indazoles--chemical synthesis
Indoles--chemical synthesis
Mice
Mice, SCID
Models, Molecular
Protein Serine-Threonine Kinases--antagonists & inhibitors
Stereoisomerism
Structure-Activity Relationship
Transplantation, Heterologous