Yang, Christine

Discovery of novel oxazolidinedione derivatives as potent and selective mineralocorticoid receptor antagonists. [electronic resource] - Bioorganic & medicinal chemistry letters Aug 2013 - 4388-92 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2013.05.077 doi


Animals
Binding Sites
Drug Evaluation, Preclinical
Half-Life
Humans
Microsomes--metabolism
Mineralocorticoid Receptor Antagonists--chemical synthesis
Molecular Docking Simulation
Oxazoles--chemical synthesis
Protein Structure, Tertiary
Rats
Receptors, Mineralocorticoid--chemistry
Structure-Activity Relationship