Design, synthesis and evaluation of inhibitor of apoptosis protein (IAP) antagonists that are highly selective for the BIR2 domain of XIAP. [electronic resource]
- Bioorganic & medicinal chemistry letters Jul 2013
- 4253-7 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1464-3405
10.1016/j.bmcl.2013.04.096 doi
Binding Sites Biomimetic Materials--chemical synthesis Cell Line, Tumor Cell Survival Drug Design Drug Resistance, Neoplasm--drug effects Humans Molecular Docking Simulation Oligopeptides--chemical synthesis Protein Binding Protein Structure, Tertiary Structure-Activity Relationship TNF-Related Apoptosis-Inducing Ligand--pharmacology X-Linked Inhibitor of Apoptosis Protein--antagonists & inhibitors