Niphakis, Micah J

Evaluation of NHS carbamates as a potent and selective class of endocannabinoid hydrolase inhibitors. [electronic resource] - ACS chemical neuroscience Sep 2013 - 1322-32 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

1948-7193

10.1021/cn400116z doi


Amidohydrolases--antagonists & inhibitors
Animals
Blood Glucose--analysis
Brain--drug effects
Carbamates--chemical synthesis
Diabetes Mellitus, Type 2--blood
Diabetic Neuropathies--blood
Drug Evaluation, Preclinical
Endocannabinoids--metabolism
HEK293 Cells
Humans
Hyperalgesia--drug therapy
Insulin--blood
Liver--drug effects
Male
Mice
Molecular Structure
Monoacylglycerol Lipases--antagonists & inhibitors
Nociception--drug effects
Rats
Rats, Sprague-Dawley
Species Specificity
Structure-Activity Relationship
Succinimides--chemistry