Zhou, Binhua

Deubiquitinase inhibition of 19S regulatory particles by 4-arylidene curcumin analog AC17 causes NF-κB inhibition and p53 reactivation in human lung cancer cells. [electronic resource] - Molecular cancer therapeutics Aug 2013 - 1381-92 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1538-8514

10.1158/1535-7163.MCT-12-1057 doi


Animals
Cell Line, Tumor
Cell Proliferation--drug effects
Curcumin--analogs & derivatives
Disease Models, Animal
Enzyme Activation--drug effects
Enzyme Inhibitors--pharmacology
Female
Humans
Lung Neoplasms--drug therapy
NF-kappa B--antagonists & inhibitors
Proteasome Endopeptidase Complex--metabolism
Proteasome Inhibitors--pharmacology
Proteolysis--drug effects
Tumor Burden--drug effects
Tumor Suppressor Protein p53--agonists
Ubiquitin-Specific Proteases--antagonists & inhibitors
Ubiquitination--drug effects
Xenograft Model Antitumor Assays