Discovery of a highly potent, nonabsorbable apical sodium-dependent bile acid transporter inhibitor (GSK2330672) for treatment of type 2 diabetes. [electronic resource]
- Journal of medicinal chemistry Jun 2013
- 5094-114 p. digital
Publication Type: Journal Article
1520-4804
10.1021/jm400459m doi
Animals Bile Acids and Salts--metabolism Diabetes Mellitus, Type 2--drug therapy Dogs Drug Discovery Drug Stability HEK293 Cells Humans Hypoglycemic Agents--chemistry Male Methylamines--chemistry Mice Organic Anion Transporters, Sodium-Dependent--antagonists & inhibitors Rats Solubility Symporters--antagonists & inhibitors Thiazepines--chemistry