Wu, Yulin

Discovery of a highly potent, nonabsorbable apical sodium-dependent bile acid transporter inhibitor (GSK2330672) for treatment of type 2 diabetes. [electronic resource] - Journal of medicinal chemistry Jun 2013 - 5094-114 p. digital

Publication Type: Journal Article

1520-4804

10.1021/jm400459m doi


Animals
Bile Acids and Salts--metabolism
Diabetes Mellitus, Type 2--drug therapy
Dogs
Drug Discovery
Drug Stability
HEK293 Cells
Humans
Hypoglycemic Agents--chemistry
Male
Methylamines--chemistry
Mice
Organic Anion Transporters, Sodium-Dependent--antagonists & inhibitors
Rats
Solubility
Symporters--antagonists & inhibitors
Thiazepines--chemistry