Effects of Rifampin, a potent inducer of drug-metabolizing enzymes and an inhibitor of OATP1B1/3 transport, on the single dose pharmacokinetics of anacetrapib. [electronic resource]
- Journal of clinical pharmacology Jul 2013
- 746-52 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1552-4604
10.1002/jcph.97 doi
Adult Area Under Curve Cytochrome P-450 CYP3A--metabolism Drug Interactions Female Humans Inactivation, Metabolic Liver-Specific Organic Anion Transporter 1 Male Middle Aged Organic Anion Transporters--antagonists & inhibitors Organic Anion Transporters, Sodium-Independent--antagonists & inhibitors Oxazolidinones--administration & dosage Rifampin--adverse effects Solute Carrier Organic Anion Transporter Family Member 1B3 Young Adult