Synthesis of pyrazolo[1,5-a]pyrimidine linked aminobenzothiazole conjugates as potential anticancer agents. [electronic resource]
- Bioorganic & medicinal chemistry letters Jun 2013
- 3208-15 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1464-3405
10.1016/j.bmcl.2013.03.129 doi
Antineoplastic Agents--chemical synthesis Apoptosis--drug effects Benzothiazoles--chemistry CDC2 Protein Kinase--metabolism Caspase 3--metabolism Cell Line, Tumor DNA Fragmentation--drug effects Drug Screening Assays, Antitumor G2 Phase Cell Cycle Checkpoints--drug effects Humans M Phase Cell Cycle Checkpoints--drug effects Pyrazoles--chemistry Pyrimidines--chemistry