Bentz, Joe

Variability in P-glycoprotein inhibitory potency (IC₅₀) using various in vitro experimental systems: implications for universal digoxin drug-drug interaction risk assessment decision criteria. [electronic resource] - Drug metabolism and disposition: the biological fate of chemicals Jul 2013 - 1347-66 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural

1521-009X

10.1124/dmd.112.050500 doi


ATP Binding Cassette Transporter, Subfamily B, Member 1--antagonists & inhibitors
Animals
Biological Transport
Caco-2 Cells
Digoxin--pharmacokinetics
Dogs
Drug Interactions
Humans
Inhibitory Concentration 50
LLC-PK1 Cells
Principal Component Analysis
Risk Assessment
Swine