Variability in P-glycoprotein inhibitory potency (IC₅₀) using various in vitro experimental systems: implications for universal digoxin drug-drug interaction risk assessment decision criteria. [electronic resource]
- Drug metabolism and disposition: the biological fate of chemicals Jul 2013
- 1347-66 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural
1521-009X
10.1124/dmd.112.050500 doi
ATP Binding Cassette Transporter, Subfamily B, Member 1--antagonists & inhibitors Animals Biological Transport Caco-2 Cells Digoxin--pharmacokinetics Dogs Drug Interactions Humans Inhibitory Concentration 50 LLC-PK1 Cells Principal Component Analysis Risk Assessment Swine