Takusagawa, Shin
Intestinal absorption mechanism of mirabegron, a potent and selective β₃-adrenoceptor agonist: involvement of human efflux and/or influx transport systems. [electronic resource]
- Molecular pharmaceutics May 2013
- 1783-94 p. digital
Publication Type: Journal Article
ISSN: 1543-8392
Standard No.: 10.1021/mp300582s doi
Subjects--Topical Terms: ATP Binding Cassette Transporter, Subfamily B, Member 1--metabolism ATP Binding Cassette Transporter, Subfamily G, Member 2 ATP-Binding Cassette Transporters--metabolism Acetanilides--pharmacokinetics Adrenergic beta-3 Receptor Agonists--pharmacokinetics Animals Biological Availability Biological Transport, Active Caco-2 Cells Cell Membrane Permeability Female HEK293 Cells Humans Hydrogen-Ion Concentration Intestinal Absorption--physiology LLC-PK1 Cells Neoplasm Proteins--metabolism Oocytes--metabolism Organic Anion Transporters--metabolism Peptide Transporter 1 Recombinant Proteins--metabolism Swine Symporters--metabolism Thiazoles--pharmacokinetics Urinary Bladder, Overactive--drug therapy Xenopus laevis