Takusagawa, Shin

Intestinal absorption mechanism of mirabegron, a potent and selective β₃-adrenoceptor agonist: involvement of human efflux and/or influx transport systems. [electronic resource] - Molecular pharmaceutics May 2013 - 1783-94 p. digital

Publication Type: Journal Article

1543-8392

10.1021/mp300582s doi


ATP Binding Cassette Transporter, Subfamily B, Member 1--metabolism
ATP Binding Cassette Transporter, Subfamily G, Member 2
ATP-Binding Cassette Transporters--metabolism
Acetanilides--pharmacokinetics
Adrenergic beta-3 Receptor Agonists--pharmacokinetics
Animals
Biological Availability
Biological Transport, Active
Caco-2 Cells
Cell Membrane Permeability
Female
HEK293 Cells
Humans
Hydrogen-Ion Concentration
Intestinal Absorption--physiology
LLC-PK1 Cells
Neoplasm Proteins--metabolism
Oocytes--metabolism
Organic Anion Transporters--metabolism
Peptide Transporter 1
Recombinant Proteins--metabolism
Swine
Symporters--metabolism
Thiazoles--pharmacokinetics
Urinary Bladder, Overactive--drug therapy
Xenopus laevis