GC-targeted C8-linked pyrrolobenzodiazepine-biaryl conjugates with femtomolar in vitro cytotoxicity and in vivo antitumor activity in mouse models. [electronic resource]
- Journal of medicinal chemistry Apr 2013
- 2911-35 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1520-4804
10.1021/jm301882a doi
Animals Antineoplastic Agents--pharmacology Benzodiazepines--chemistry Cell Line, Tumor Disease Models, Animal Drug Screening Assays, Antitumor Fluorescence Resonance Energy Transfer GC Rich Sequence Humans In Vitro Techniques Magnetic Resonance Spectroscopy Mice Models, Molecular Molecular Structure NF-kappa B--antagonists & inhibitors Spectrometry, Mass, Electrospray Ionization