Rahman, Khondaker M

GC-targeted C8-linked pyrrolobenzodiazepine-biaryl conjugates with femtomolar in vitro cytotoxicity and in vivo antitumor activity in mouse models. [electronic resource] - Journal of medicinal chemistry Apr 2013 - 2911-35 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1520-4804

10.1021/jm301882a doi


Animals
Antineoplastic Agents--pharmacology
Benzodiazepines--chemistry
Cell Line, Tumor
Disease Models, Animal
Drug Screening Assays, Antitumor
Fluorescence Resonance Energy Transfer
GC Rich Sequence
Humans
In Vitro Techniques
Magnetic Resonance Spectroscopy
Mice
Models, Molecular
Molecular Structure
NF-kappa B--antagonists & inhibitors
Spectrometry, Mass, Electrospray Ionization