Gajula, Praveen Kumar

A synthetic dolastatin 10 analogue suppresses microtubule dynamics, inhibits cell proliferation, and induces apoptotic cell death. [electronic resource] - Journal of medicinal chemistry Mar 2013 - 2235-45 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1520-4804

10.1021/jm3009629 doi


Antineoplastic Agents--chemical synthesis
Apoptosis--drug effects
Caspase 3--metabolism
Cell Proliferation--drug effects
Colchicine--pharmacology
Depsipeptides--chemical synthesis
Drug Interactions
Drug Resistance, Neoplasm--drug effects
GTP Phosphohydrolases--metabolism
HeLa Cells
Humans
JNK Mitogen-Activated Protein Kinases--metabolism
Kinetochores--drug effects
MCF-7 Cells
Microtubules--drug effects
Mitosis--drug effects
Protein Multimerization--drug effects
Protein Structure, Quaternary
Tubulin--chemistry
Vinblastine--pharmacology