Substrate and inhibitor-induced dimerization and cooperativity in caspase-1 but not caspase-3. [electronic resource]
- The Journal of biological chemistry Apr 2013
- 9971-9981 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, Non-P.H.S.
1083-351X
10.1074/jbc.M112.426460 doi
Allosteric Site Amino Acid Chloromethyl Ketones--chemistry Area Under Curve Biophysics--methods Caspase 1--metabolism Caspase 3--metabolism Caspases--metabolism Catalytic Domain Dimerization Enzyme Inhibitors--pharmacology Gene Expression Regulation, Enzymologic Humans Inflammation Kinetics Models, Molecular Molecular Conformation Protein Binding Protein Conformation Substrate Specificity Ultracentrifugation