Wang, Zhi-Peng

The effect of absolute configuration on activity, subtype selectivity (M3/M2) of 3α-acyloxy-6β-acetoxyltropane derivatives as muscarinic M3 receptor antagonists. [electronic resource] - Bioorganic & medicinal chemistry Mar 2013 - 1234-9 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1464-3391

10.1016/j.bmc.2012.12.052 doi


Animals
Female
Guinea Pigs
Heart Atria--drug effects
Ileum--drug effects
Male
Muscarinic Antagonists--chemical synthesis
Radioligand Assay
Rats
Receptor, Muscarinic M2--antagonists & inhibitors
Receptor, Muscarinic M3--antagonists & inhibitors
Structure-Activity Relationship
Tropanes--chemical synthesis