Colabufo, Nicola A

Naphthalenyl derivatives for hitting P-gp/MRP1/BCRP transporters. [electronic resource] - Bioorganic & medicinal chemistry Mar 2013 - 1324-32 p. digital

Publication Type: Journal Article

1464-3391

10.1016/j.bmc.2012.12.021 doi


ATP Binding Cassette Transporter, Subfamily B, Member 1--antagonists & inhibitors
ATP-Binding Cassette Transporters--antagonists & inhibitors
Animals
Caco-2 Cells
Cell Proliferation--drug effects
Dogs
Drug Carriers--chemistry
Humans
Madin Darby Canine Kidney Cells
Multidrug Resistance-Associated Proteins--antagonists & inhibitors
Naphthalenes--chemical synthesis
Oxazoles--chemistry
Rhodamine 123--chemistry
Structure-Activity Relationship
Substrate Specificity
Thiazoles--chemistry