Colabufo, Nicola A
Naphthalenyl derivatives for hitting P-gp/MRP1/BCRP transporters. [electronic resource]
- Bioorganic & medicinal chemistry Mar 2013
- 1324-32 p. digital
Publication Type: Journal Article
ISSN: 1464-3391
Standard No.: 10.1016/j.bmc.2012.12.021 doi
Subjects--Topical Terms: ATP Binding Cassette Transporter, Subfamily B, Member 1--antagonists & inhibitors ATP-Binding Cassette Transporters--antagonists & inhibitors Animals Caco-2 Cells Cell Proliferation--drug effects Dogs Drug Carriers--chemistry Humans Madin Darby Canine Kidney Cells Multidrug Resistance-Associated Proteins--antagonists & inhibitors Naphthalenes--chemical synthesis Oxazoles--chemistry Rhodamine 123--chemistry Structure-Activity Relationship Substrate Specificity Thiazoles--chemistry