Distinct CCK-2 receptor conformations associated with β-arrestin-2 recruitment or phospholipase-C activation revealed by a biased antagonist. [electronic resource]
- Journal of the American Chemical Society Feb 2013
- 2560-73 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1520-5126
10.1021/ja308784w doi
Adamantane--analogs & derivatives Arrestins--chemistry Binding Sites Enzyme Activation--drug effects Humans Microscopy, Confocal Models, Molecular Molecular Structure Mutation Phenylurea Compounds--pharmacology Protein Conformation Receptor, Cholecystokinin B--antagonists & inhibitors Signal Transduction Type C Phospholipases--chemistry Up-Regulation beta-Arrestin 2 beta-Arrestins