Chou, Tsui-Fen

Structure-activity relationship study reveals ML240 and ML241 as potent and selective inhibitors of p97 ATPase. [electronic resource] - ChemMedChem Feb 2013 - 297-312 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

1860-7187

10.1002/cmdc.201200520 doi


Adenosine Triphosphatases--antagonists & inhibitors
Antineoplastic Agents--chemistry
Autophagy--drug effects
Benzimidazoles--chemistry
Benzoxazines
Caspases--metabolism
Cell Line, Tumor
Cell Proliferation--drug effects
Endoplasmic Reticulum-Associated Degradation--drug effects
Humans
Neoplasms--drug therapy
Nuclear Proteins--antagonists & inhibitors
Proteasome Endopeptidase Complex--metabolism
Proteasome Inhibitors--pharmacology
Quinazolines--chemistry
Structure-Activity Relationship
Ubiquitin--metabolism