TY  - GEN
AU  - Fujishiro,Shinya
AU  - Dodo,Kosuke
AU  - Iwasa,Eriko
AU  - Teng,Yuou
AU  - Sohtome,Yoshihiro
AU  - Hamashima,Yoshitaka
AU  - Ito,Akihiro
AU  - Yoshida,Minoru
AU  - Sodeoka,Mikiko
TI  - Epidithiodiketopiperazine as a pharmacophore for protein lysine methyltransferase G9a inhibitors: reducing cytotoxicity by structural simplification
SN  - 1464-3405
PY  - 2013///0625
KW  - Cell Survival
KW  - drug effects
KW  - Chaetomium
KW  - chemistry
KW  - Diketopiperazines
KW  - chemical synthesis
KW  - Enzyme Inhibitors
KW  - HL-60 Cells
KW  - Histone-Lysine N-Methyltransferase
KW  - antagonists & inhibitors
KW  - Humans
KW  - Molecular Structure
KW  - Piperazines
KW  - Structure-Activity Relationship
KW  - Thioredoxin-Disulfide Reductase
KW  - metabolism
N1  - Publication Type: Journal Article; Research Support, Non-U.S. Gov't
UR  - https://doi.org/10.1016/j.bmcl.2012.11.087
ER  -