Budke, Brian

An optimized RAD51 inhibitor that disrupts homologous recombination without requiring Michael acceptor reactivity. [electronic resource] - Journal of medicinal chemistry Jan 2013 - 254-63 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural

1520-4804

10.1021/jm301565b doi


Binding Sites
DNA--chemistry
DNA Repair--drug effects
HEK293 Cells
Homologous Recombination--drug effects
Humans
Maleimides--chemical synthesis
Morpholines--chemical synthesis
Protein Binding
Pyrroles--chemistry
Rad51 Recombinase--antagonists & inhibitors
Structure-Activity Relationship