TY  - GEN
AU  - Lee,Kijae
AU  - Pham,Van Chung
AU  - Choi,Min Ji
AU  - Kim,Kyung Ju
AU  - Lee,Kyung-Tae
AU  - Han,Seong-Gu
AU  - Yu,Yeon Gyu
AU  - Lee,Jae Yeol
TI  - Fragment-based discovery of novel and selective mPGES-1 inhibitors Part 1: identification of sulfonamido-1,2,3-triazole-4,5-dicarboxylic acid
SN  - 1464-3405
PY  - 2013///0528
KW  - Binding Sites
KW  - Catalytic Domain
KW  - Crystallography, X-Ray
KW  - Dicarboxylic Acids
KW  - chemical synthesis
KW  - Drug Design
KW  - Drug Evaluation, Preclinical
KW  - Enzyme Inhibitors
KW  - Humans
KW  - Intramolecular Oxidoreductases
KW  - antagonists & inhibitors
KW  - Microsomes
KW  - enzymology
KW  - Molecular Docking Simulation
KW  - Prostaglandin-E Synthases
KW  - Protein Binding
KW  - Sulfonamides
KW  - Thermodynamics
KW  - Triazoles
N1  - Publication Type: Journal Article; Research Support, Non-U.S. Gov't
UR  - https://doi.org/10.1016/j.bmcl.2012.11.019
ER  -