Structure-activity relationships and blood distribution of antiplasmodial aminopeptidase-1 inhibitors. [electronic resource]
- Journal of medicinal chemistry Dec 2012
- 10909-17 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1520-4804
10.1021/jm301506h doi
Aminopeptidases--antagonists & inhibitors Animals Antimalarials--blood Cell Line Drug Resistance Female Humans Malaria--drug therapy Malonates--blood Metalloproteases--antagonists & inhibitors Mice Molecular Docking Simulation Plasmodium berghei Plasmodium falciparum--drug effects Protein Binding Protozoan Proteins--antagonists & inhibitors Rats Solubility Stereoisomerism Structure-Activity Relationship Tissue Distribution Zinc