Choi, Eunhyun

Property-based optimization of hydroxamate-based γ-lactam HDAC inhibitors to improve their metabolic stability and pharmacokinetic profiles. [electronic resource] - Journal of medicinal chemistry Dec 2012 - 10766-70 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1520-4804

10.1021/jm3009376 doi


Histone Deacetylase Inhibitors--chemistry
Hydroxamic Acids--chemistry
Lactams--chemistry
Magnetic Resonance Spectroscopy