Property-based optimization of hydroxamate-based γ-lactam HDAC inhibitors to improve their metabolic stability and pharmacokinetic profiles. [electronic resource]
- Journal of medicinal chemistry Dec 2012
- 10766-70 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1520-4804
10.1021/jm3009376 doi
Histone Deacetylase Inhibitors--chemistry Hydroxamic Acids--chemistry Lactams--chemistry Magnetic Resonance Spectroscopy