TY  - GEN
AU  - Rodriguez,Alice L
AU  - Zhou,Ya
AU  - Williams,Richard
AU  - Weaver,C David
AU  - Vinson,Paige N
AU  - Dawson,Eric S
AU  - Steckler,Thomas
AU  - Lavreysen,Hilde
AU  - Mackie,Claire
AU  - Bartolomé,José M
AU  - Macdonald,Gregor J
AU  - Daniels,J Scott
AU  - Niswender,Colleen M
AU  - Jones,Carrie K
AU  - Conn,P Jeffrey
AU  - Lindsley,Craig W
AU  - Stauffer,Shaun R
TI  - Discovery and SAR of a novel series of non-MPEP site mGlu₅ PAMs based on an aryl glycine sulfonamide scaffold
SN  - 1464-3405
PY  - 2013///0520
KW  - Allosteric Regulation
KW  - drug effects
KW  - Animals
KW  - Binding Sites
KW  - Dose-Response Relationship, Drug
KW  - Drug Discovery
KW  - Glycine
KW  - analogs & derivatives
KW  - Humans
KW  - Models, Molecular
KW  - Molecular Structure
KW  - Rats
KW  - Receptor, Metabotropic Glutamate 5
KW  - Receptors, Metabotropic Glutamate
KW  - chemistry
KW  - Structure-Activity Relationship
KW  - Sulfonamides
KW  - chemical synthesis
N1  - Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
UR  - https://doi.org/10.1016/j.bmcl.2012.10.068
ER  -