Rodriguez, Alice L

Discovery and SAR of a novel series of non-MPEP site mGlu₅ PAMs based on an aryl glycine sulfonamide scaffold. [electronic resource] - Bioorganic & medicinal chemistry letters Dec 2012 - 7388-92 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

1464-3405

10.1016/j.bmcl.2012.10.068 doi


Allosteric Regulation--drug effects
Animals
Binding Sites--drug effects
Dose-Response Relationship, Drug
Drug Discovery
Glycine--analogs & derivatives
Humans
Models, Molecular
Molecular Structure
Rats
Receptor, Metabotropic Glutamate 5
Receptors, Metabotropic Glutamate--chemistry
Structure-Activity Relationship
Sulfonamides--chemical synthesis