Cheung, Adrian Wai-Hing

7-Phenyl-pyrido[2,3-d]pyrimidine-2,4-diamines: novel and highly selective protein tyrosine phosphatase 1B inhibitors. [electronic resource] - Bioorganic & medicinal chemistry letters Dec 2012 - 7518-22 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2012.10.035 doi


Animals
Diamines--chemical synthesis
Dose-Response Relationship, Drug
Enzyme Inhibitors--administration & dosage
Humans
Mice
Mice, Inbred C57BL
Molecular Structure
Protein Tyrosine Phosphatase, Non-Receptor Type 1--antagonists & inhibitors
Pyrimidines--chemical synthesis
Structure-Activity Relationship