7-Phenyl-pyrido[2,3-d]pyrimidine-2,4-diamines: novel and highly selective protein tyrosine phosphatase 1B inhibitors. [electronic resource]
- Bioorganic & medicinal chemistry letters Dec 2012
- 7518-22 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2012.10.035 doi
Animals Diamines--chemical synthesis Dose-Response Relationship, Drug Enzyme Inhibitors--administration & dosage Humans Mice Mice, Inbred C57BL Molecular Structure Protein Tyrosine Phosphatase, Non-Receptor Type 1--antagonists & inhibitors Pyrimidines--chemical synthesis Structure-Activity Relationship