TY - GEN AU - Angelini,Alessandro AU - Morales-Sanfrutos,Julia AU - Diderich,Philippe AU - Chen,Shiyu AU - Heinis,Christian TI - Bicyclization and tethering to albumin yields long-acting peptide antagonists SN - 1520-4804 PY - 2013///0205 KW - Animals KW - Bridged Bicyclo Compounds KW - blood KW - Cyclization KW - Female KW - Mice KW - Mice, Inbred BALB C KW - Models, Molecular KW - Molecular Structure KW - Peptides, Cyclic KW - Serum Albumin KW - metabolism KW - Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization KW - Structure-Activity Relationship KW - Urokinase-Type Plasminogen Activator KW - antagonists & inhibitors N1 - Publication Type: Journal Article; Research Support, Non-U.S. Gov't UR - https://doi.org/10.1021/jm301276e ER -