Characterisation of the roles of ABCB1, ABCC1, ABCC2 and ABCG2 in the transport and pharmacokinetics of actinomycin D in vitro and in vivo. [electronic resource]
- Biochemical pharmacology Jan 2013
- 29-37 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1873-2968
10.1016/j.bcp.2012.10.004 doi
ATP Binding Cassette Transporter, Subfamily B ATP Binding Cassette Transporter, Subfamily B, Member 1--genetics ATP Binding Cassette Transporter, Subfamily G, Member 2 ATP-Binding Cassette Transporters--metabolism Animals Antibiotics, Antineoplastic--blood Biological Transport Cell Proliferation--drug effects Dactinomycin--blood Dogs Doxorubicin--pharmacokinetics Humans Madin Darby Canine Kidney Cells Mice Mice, Knockout Multidrug Resistance-Associated Protein 2 Multidrug Resistance-Associated Proteins--genetics Neoplasm Proteins--metabolism Tissue Distribution