Zhang, Peng

Design, synthesis and biological evaluation of benzothiazepinones (BTZs) as novel non-ATP competitive inhibitors of glycogen synthase kinase-3β (GSK-3β). [electronic resource] - European journal of medicinal chemistry Mar 2013 - 95-103 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1768-3254

10.1016/j.ejmech.2012.09.021 doi


Benzazepines--chemical synthesis
Binding, Competitive--drug effects
Crystallography, X-Ray
Dose-Response Relationship, Drug
Drug Design
Glycogen Synthase Kinase 3--antagonists & inhibitors
Glycogen Synthase Kinase 3 beta
Humans
Models, Molecular
Molecular Structure
Protein Kinase Inhibitors--chemical synthesis
Recombinant Proteins--metabolism
Structure-Activity Relationship