Provins, Laurent <br/><br/>
Lead optimization of thiazolo[5,4-c]piperidines: 3-cyclobutoxy linker as a key spacer for H(3)R inverse agonists.  [electronic resource] 

 -  ChemMedChem  Dec 2012 
 - 2087-92 p.  digital 
<br/><br/> Publication Type: Journal Article; Research Support, Non-U.S. Gov't 
<br/><br/><label>ISSN: </label>1860-7187 
<br/><br/><label>Standard No.: </label>10.1002/cmdc.201200406  doi 
<br/><br/><label>Subjects--Topical Terms: </label><br/>Animals<br/>Benzamides--chemistry<br/>Caco-2 Cells<br/>Histamine Agonists--chemistry<br/>Humans<br/>Male<br/>Piperidines--chemistry<br/>Rats<br/>Rats, Wistar<br/>Receptors, Histamine H3--metabolism<br/>Structure-Activity Relationship<br/>Thiazoles--chemistry<br/>Trans-Activators--metabolism<br/>Transcriptional Regulator ERG