Kung, Charles
Small molecule activation of PKM2 in cancer cells induces serine auxotrophy. [electronic resource]
- Chemistry & biology Sep 2012
- 1187-98 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1879-1301
10.1016/j.chembiol.2012.07.021 doi
Allosteric Site--drug effects
Carrier Proteins--metabolism
Cell Proliferation--drug effects
Dose-Response Relationship, Drug
Humans
Membrane Proteins--metabolism
Models, Molecular
Molecular Structure
Serine--metabolism
Small Molecule Libraries--chemical synthesis
Structure-Activity Relationship
Thyroid Hormones--metabolism
Tumor Cells, Cultured
Thyroid Hormone-Binding Proteins