Meng, Fei

Structure-based discovery of highly selective phosphodiesterase-9A inhibitors and implications for inhibitor design. [electronic resource] - Journal of medicinal chemistry Oct 2012 - 8549-58 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

1520-4804

10.1021/jm301189c doi


3',5'-Cyclic-AMP Phosphodiesterases--chemistry
Catalytic Domain
Crystallography, X-Ray
Drug Design
Molecular Docking Simulation
Phosphodiesterase Inhibitors--chemical synthesis
Pyrazoles--chemical synthesis
Pyrimidines--chemical synthesis
Structure-Activity Relationship