The inhibition of the potassium channel TASK-1 in rat cardiac muscle by endothelin-1 is mediated by phospholipase C. [electronic resource]
- Cardiovascular research Jan 2013
- 97-105 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1755-3245
10.1093/cvr/cvs285 doi
Action Potentials Animals CHO Cells Cricetinae Cricetulus Endothelin-1--pharmacology Enzyme Activation Enzyme Inhibitors--pharmacology Hydrogen-Ion Concentration Hydrolysis Ion Channel Gating Kinetics Microscopy, Fluorescence Microscopy, Interference Myocytes, Cardiac--drug effects Nerve Tissue Proteins Patch-Clamp Techniques Phosphatidylinositol 4,5-Diphosphate--metabolism Potassium Channel Blockers--pharmacology Potassium Channels, Tandem Pore Domain--antagonists & inhibitors Rats Receptor, Endothelin A--genetics Signal Transduction--drug effects Transfection Type C Phospholipases--antagonists & inhibitors