Fuchs, Ines
Effect of the CYP3A inhibitor ketoconazole on the PXR-mediated induction of CYP3A activity. [electronic resource]
- European journal of clinical pharmacology Mar 2013
- 507-13 p. digital
Publication Type: Comparative Study; Journal Article; Randomized Controlled Trial
ISSN: 1432-1041
Standard No.: 10.1007/s00228-012-1388-1 doi
Subjects--Topical Terms: Adult Area Under Curve Biotransformation Cross-Over Studies Cytochrome P-450 CYP3A--biosynthesis Cytochrome P-450 CYP3A Inhibitors Drug Administration Schedule Drug Interactions Enzyme Induction Enzyme Inhibitors--administration & dosage Germany Humans Hydroxylation Hypericum Ketoconazole--administration & dosage Male Metabolic Clearance Rate Midazolam--administration & dosage Middle Aged Plant Extracts--administration & dosage Plants, Medicinal Pregnane X Receptor Receptors, Steroid--drug effects Substrate Specificity Transcription, Genetic--drug effects Young Adult