Erickson, J

Design, activity, and 2.8 A crystal structure of a C2 symmetric inhibitor complexed to HIV-1 protease. [electronic resource] - Science (New York, N.Y.) Aug 1990 - 527-33 p. digital

Publication Type: Journal Article; Research Support, U.S. Gov't, P.H.S.

0036-8075

10.1126/science.2200122 doi


Amino Acid Sequence
Binding Sites
Drug Design
Endopeptidases--metabolism
Gene Products, pol--metabolism
HIV Protease
HIV-1--enzymology
Kinetics
Models, Molecular
Molecular Sequence Data
Protease Inhibitors--pharmacology
Protein Conformation
Sugar Alcohols--pharmacology
Valine--analogs & derivatives