Design, activity, and 2.8 A crystal structure of a C2 symmetric inhibitor complexed to HIV-1 protease. [electronic resource]
- Science (New York, N.Y.) Aug 1990
- 527-33 p. digital
Publication Type: Journal Article; Research Support, U.S. Gov't, P.H.S.
0036-8075
10.1126/science.2200122 doi
Amino Acid Sequence Binding Sites Drug Design Endopeptidases--metabolism Gene Products, pol--metabolism HIV Protease HIV-1--enzymology Kinetics Models, Molecular Molecular Sequence Data Protease Inhibitors--pharmacology Protein Conformation Sugar Alcohols--pharmacology Valine--analogs & derivatives