A selective ATP-binding cassette subfamily G member 2 efflux inhibitor revealed via high-throughput flow cytometry. [electronic resource]
- Journal of biomolecular screening Jan 2013
- 26-38 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1552-454X
10.1177/1087057112456875 doi
ATP Binding Cassette Transporter, Subfamily B ATP Binding Cassette Transporter, Subfamily B, Member 1--antagonists & inhibitors ATP Binding Cassette Transporter, Subfamily G, Member 2 ATP-Binding Cassette Transporters--antagonists & inhibitors Animals Antineoplastic Agents--pharmacology Cell Line Drug Resistance, Neoplasm Flow Cytometry High-Throughput Screening Assays Humans Inhibitory Concentration 50 Mice Mice, SCID Neoplasm Proteins--antagonists & inhibitors Pyrazoles--pharmacology Pyrimidines--pharmacology Small Molecule Libraries Structure-Activity Relationship Tumor Burden--drug effects Xenograft Model Antitumor Assays