Strouse, J Jacob

A selective ATP-binding cassette subfamily G member 2 efflux inhibitor revealed via high-throughput flow cytometry. [electronic resource] - Journal of biomolecular screening Jan 2013 - 26-38 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1552-454X

10.1177/1087057112456875 doi


ATP Binding Cassette Transporter, Subfamily B
ATP Binding Cassette Transporter, Subfamily B, Member 1--antagonists & inhibitors
ATP Binding Cassette Transporter, Subfamily G, Member 2
ATP-Binding Cassette Transporters--antagonists & inhibitors
Animals
Antineoplastic Agents--pharmacology
Cell Line
Drug Resistance, Neoplasm
Flow Cytometry
High-Throughput Screening Assays
Humans
Inhibitory Concentration 50
Mice
Mice, SCID
Neoplasm Proteins--antagonists & inhibitors
Pyrazoles--pharmacology
Pyrimidines--pharmacology
Small Molecule Libraries
Structure-Activity Relationship
Tumor Burden--drug effects
Xenograft Model Antitumor Assays