Hua, Zihao

2-Phenylamino-6-cyano-1H-benzimidazole-based isoform selective casein kinase 1 gamma (CK1γ) inhibitors. [electronic resource] - Bioorganic & medicinal chemistry letters Sep 2012 - 5392-5 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2012.07.046 doi


Animals
Benzimidazoles--chemistry
Binding Sites
Casein Kinase I--antagonists & inhibitors
Humans
Mice
Models, Molecular
Protein Isoforms--antagonists & inhibitors
Protein Kinase Inhibitors--chemistry
Rats
Structure-Activity Relationship
beta Catenin--metabolism