Blockade of STAT3 activation by sorafenib derivatives through enhancing SHP-1 phosphatase activity. [electronic resource]
- European journal of medicinal chemistry Sep 2012
- 220-7 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1768-3254
10.1016/j.ejmech.2012.07.023 doi
Animals Benzenesulfonates--chemistry Cell Line, Tumor Dose-Response Relationship, Drug Down-Regulation--drug effects Humans Male Mice Mice, Nude Niacinamide--analogs & derivatives Phenylurea Compounds Phosphoproteins--metabolism Protein Kinase Inhibitors--analogs & derivatives Protein Kinases--metabolism Protein Tyrosine Phosphatase, Non-Receptor Type 6--metabolism Pyridines--chemistry STAT3 Transcription Factor--metabolism Sorafenib Xenograft Model Antitumor Assays