TY - GEN AU - Liddle,John AU - Bamborough,Paul AU - Barker,Michael D AU - Campos,Sebastien AU - Chung,Chun-Wa AU - Cousins,Rick P C AU - Faulder,Paul AU - Heathcote,Michelle L AU - Hobbs,Heather AU - Holmes,Duncan S AU - Ioannou,Chris AU - Ramirez-Molina,Cesar AU - Morse,Mary A AU - Osborn,Ruth AU - Payne,Jeremy J AU - Pritchard,John M AU - Rumsey,William L AU - Tape,Daniel T AU - Vicentini,Giorgia AU - Whitworth,Caroline AU - Williamson,Rick A TI - 4-Phenyl-7-azaindoles as potent, selective and bioavailable IKK2 inhibitors demonstrating good in vivo efficacy SN - 1464-3405 PY - 2012///1130 KW - Animals KW - Biological Availability KW - Disease Models, Animal KW - Half-Life KW - Humans KW - I-kappa B Kinase KW - antagonists & inhibitors KW - Indoles KW - chemical synthesis KW - Lung KW - metabolism KW - Neutrophils KW - immunology KW - Protein Kinase Inhibitors KW - Rats KW - Structure-Activity Relationship N1 - Publication Type: Journal Article UR - https://doi.org/10.1016/j.bmcl.2012.06.065 ER -