Liddle, John 4-Phenyl-7-azaindoles as potent, selective and bioavailable IKK2 inhibitors demonstrating good in vivo efficacy. [electronic resource] - Bioorganic & medicinal chemistry letters Aug 2012 - 5222-6 p. digital Publication Type: Journal Article ISSN: 1464-3405 Standard No.: 10.1016/j.bmcl.2012.06.065 doi Subjects--Topical Terms: AnimalsBiological AvailabilityDisease Models, AnimalHalf-LifeHumansI-kappa B Kinase--antagonists & inhibitorsIndoles--chemical synthesisLung--metabolismNeutrophils--immunologyProtein Kinase Inhibitors--chemical synthesisRatsStructure-Activity Relationship