Liddle, John

4-Phenyl-7-azaindoles as potent, selective and bioavailable IKK2 inhibitors demonstrating good in vivo efficacy. [electronic resource] - Bioorganic & medicinal chemistry letters Aug 2012 - 5222-6 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2012.06.065 doi


Animals
Biological Availability
Disease Models, Animal
Half-Life
Humans
I-kappa B Kinase--antagonists & inhibitors
Indoles--chemical synthesis
Lung--metabolism
Neutrophils--immunology
Protein Kinase Inhibitors--chemical synthesis
Rats
Structure-Activity Relationship