Daskalopoulos, Evangelos P

Dâ‚‚-dopaminergic receptor-linked pathways: critical regulators of CYP3A, CYP2C, and CYP2D. [electronic resource] - Molecular pharmacology Oct 2012 - 668-78 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1521-0111

10.1124/mol.112.078709 doi


Animals
Antipsychotic Agents--adverse effects
Cytochrome P-450 CYP3A--metabolism
Cytochrome P-450 Enzyme System--metabolism
Dopamine D2 Receptor Antagonists
Ethanolamines--metabolism
Forkhead Transcription Factors--physiology
Gene Expression Regulation
Hepatocytes--drug effects
Hormones--blood
In Vitro Techniques
Male
Microsomes, Liver--drug effects
Nerve Tissue Proteins--physiology
Phosphatidylinositol 3-Kinases--physiology
Phosphorylation
Proto-Oncogene Proteins c-akt--physiology
Rats
Receptors, Dopamine D2--physiology
STAT5 Transcription Factor--metabolism
Signal Transduction
Sulpiride--adverse effects