Dzierba, Carolyn D

Synthesis and structure-activity relationships of pyrido[3,2-b]pyrazin-3(4H)-ones and pteridin-7(8H)-ones as corticotropin-releasing factor-1 receptor antagonists. [electronic resource] - Bioorganic & medicinal chemistry letters Aug 2012 - 4986-9 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2012.06.034 doi


Animals
Anti-Anxiety Agents--chemical synthesis
Half-Life
Pteridines--chemical synthesis
Pyrazines--chemical synthesis
Rats
Receptors, Corticotropin-Releasing Hormone--antagonists & inhibitors
Structure-Activity Relationship
CRF Receptor, Type 1