TY - GEN AU - Mangin,Floriane AU - Dilly,Sébastien AU - Joly,Benoît AU - Scuvée-Moreau,Jacqueline AU - Evans,Jon AU - Setola,Vincent AU - Roth,Bryan L AU - Liégeois,Jean-François TI - Moderate chemical modifications of WAY-100635 improve the selectivity for 5-HT1A versus D4 receptors SN - 1464-3405 PY - 2013///0104 KW - Molecular Structure KW - Piperazines KW - chemistry KW - Pyridines KW - Receptor, Serotonin, 5-HT1A KW - metabolism KW - Receptors, Dopamine D4 KW - antagonists & inhibitors KW - Serotonin 5-HT1 Receptor Antagonists KW - Structure-Activity Relationship N1 - Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't UR - https://doi.org/10.1016/j.bmcl.2012.05.119 ER -