Majumdar, Susruta

Synthesis and evaluation of aryl-naloxamide opiate analgesics targeting truncated exon 11-associated μ opioid receptor (MOR-1) splice variants. [electronic resource] - Journal of medicinal chemistry Jul 2012 - 6352-62 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

1520-4804

10.1021/jm300305c doi


Amides--chemical synthesis
Analgesics--chemical synthesis
Animals
Behavior, Animal--drug effects
Brain--drug effects
Cell Line
Chemistry Techniques, Synthetic
Exons--genetics
Male
Mice
Opiate Alkaloids--chemical synthesis
Protein Isoforms--chemistry
Protein Structure, Tertiary
Receptors, Opioid, mu--chemistry
Structure-Activity Relationship