Shi, Qian

Antitumor agents 290. Design, synthesis, and biological evaluation of new LNCaP and PC-3 cytotoxic curcumin analogs conjugated with anti-androgens. [electronic resource] - Bioorganic & medicinal chemistry Jul 2012 - 4020-31 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

1464-3391

10.1016/j.bmc.2012.05.011 doi


Androgen Antagonists--chemistry
Anilides--chemical synthesis
Antineoplastic Agents--chemical synthesis
Cell Line, Tumor
Cell Survival--drug effects
Curcumin--analogs & derivatives
Drug Design
Flutamide--chemistry
Humans
Male
Nitriles--chemistry
Prostatic Neoplasms--drug therapy
Pseudopodia--drug effects
Structure-Activity Relationship
Tosyl Compounds--chemistry