Antimalarial activity and mechanisms of action of two novel 4-aminoquinolines against chloroquine-resistant parasites. [electronic resource]
- PloS one 2012
- e37259 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1932-6203
10.1371/journal.pone.0037259 doi
Aminoquinolines--chemistry Animals Antimalarials--chemistry Cell Line, Tumor Chloroquine Dose-Response Relationship, Drug Drug Resistance--physiology Enzyme-Linked Immunosorbent Assay Hemeproteins--antagonists & inhibitors Humans In Vitro Techniques L-Lactate Dehydrogenase--metabolism Malaria--drug therapy Mice Models, Molecular Molecular Structure Plasmodium berghei--drug effects Plasmodium falciparum--drug effects Protein Binding Protein Conformation Tetrazolium Salts Thiazoles