Enhancing chemosensitivity in ABCB1- and ABCG2-overexpressing cells and cancer stem-like cells by an Aurora kinase inhibitor CCT129202. [electronic resource]
- Molecular pharmaceutics Jul 2012
- 1971-82 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1543-8392
10.1021/mp2006714 doi
ATP Binding Cassette Transporter, Subfamily B ATP Binding Cassette Transporter, Subfamily B, Member 1--metabolism ATP Binding Cassette Transporter, Subfamily G, Member 2 ATP-Binding Cassette Transporters--metabolism Animals Antineoplastic Agents--pharmacology Aurora Kinases--antagonists & inhibitors Cell Line Cell Line, Tumor Drug Interactions Drug Resistance, Multiple--drug effects HEK293 Cells HL-60 Cells Humans Imidazoles--pharmacology MCF-7 Cells Male Mice Mice, Inbred BALB C Mice, Nude Neoplasm Proteins--metabolism Neoplastic Stem Cells--drug effects Protein Kinase Inhibitors--pharmacology Pyridines--pharmacology