Cheng, Chao

Enhancing chemosensitivity in ABCB1- and ABCG2-overexpressing cells and cancer stem-like cells by an Aurora kinase inhibitor CCT129202. [electronic resource] - Molecular pharmaceutics Jul 2012 - 1971-82 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1543-8392

10.1021/mp2006714 doi


ATP Binding Cassette Transporter, Subfamily B
ATP Binding Cassette Transporter, Subfamily B, Member 1--metabolism
ATP Binding Cassette Transporter, Subfamily G, Member 2
ATP-Binding Cassette Transporters--metabolism
Animals
Antineoplastic Agents--pharmacology
Aurora Kinases--antagonists & inhibitors
Cell Line
Cell Line, Tumor
Drug Interactions
Drug Resistance, Multiple--drug effects
HEK293 Cells
HL-60 Cells
Humans
Imidazoles--pharmacology
MCF-7 Cells
Male
Mice
Mice, Inbred BALB C
Mice, Nude
Neoplasm Proteins--metabolism
Neoplastic Stem Cells--drug effects
Protein Kinase Inhibitors--pharmacology
Pyridines--pharmacology