Davies, Christopher W

The co-crystal structure of ubiquitin carboxy-terminal hydrolase L1 (UCHL1) with a tripeptide fluoromethyl ketone (Z-VAE(OMe)-FMK). [electronic resource] - Bioorganic & medicinal chemistry letters Jun 2012 - 3900-4 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, U.S. Gov't, Non-P.H.S.

1464-3405

10.1016/j.bmcl.2012.04.124 doi


Amino Acid Chloromethyl Ketones--chemistry
Animals
Catalytic Domain
Crystallization
Crystallography, X-Ray
Humans
Models, Molecular
Oligopeptides--chemistry
Protein Binding
Protein Conformation
Substrate Specificity
Ubiquitin--chemistry
Ubiquitin Thiolesterase--chemistry