Shan, Yibing

Oncogenic mutations counteract intrinsic disorder in the EGFR kinase and promote receptor dimerization. [electronic resource] - Cell May 2012 - 860-70 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural

1097-4172

10.1016/j.cell.2012.02.063 doi


Amino Acid Sequence
Crystallography, X-Ray
ErbB Receptors--antagonists & inhibitors
Gefitinib
Humans
Lapatinib
Molecular Dynamics Simulation
Molecular Sequence Data
Neoplasms--metabolism
Point Mutation
Protein Folding
Protein Kinase Inhibitors--pharmacology
Protein Multimerization
Protein Structure, Tertiary
Quinazolines--pharmacology
Sequence Alignment
Signal Transduction