Martínez González, Sonia Identification of ETP-46321, a potent and orally bioavailable PI3K α, δ inhibitor. [electronic resource] - Bioorganic & medicinal chemistry letters May 2012 - 3460-6 p. digital Publication Type: Journal Article; Research Support, Non-U.S. Gov't ISSN: 1464-3405 Standard No.: 10.1016/j.bmcl.2012.03.090 doi Subjects--Topical Terms: Administration, OralBiological AvailabilityHumansImidazoles--administration & dosageIsoenzymes--antagonists & inhibitorsPhosphoinositide-3 Kinase InhibitorsPositron-Emission TomographyProtein Kinase Inhibitors--administration & dosagePyrazines--administration & dosageTomography, X-Ray Computed