Cowart, Marlon Pharmacological characterization of A-960656, a histamine H₃ receptor antagonist with efficacy in animal models of osteoarthritis and neuropathic pain. [electronic resource] - European journal of pharmacology Jun 2012 - 87-94 p. digital Publication Type: Journal Article ISSN: 1879-0712 Standard No.: 10.1016/j.ejphar.2012.03.048 doi Subjects--Topical Terms: AnimalsBenzothiazoles--adverse effectsCell Membrane PermeabilityCytochrome P-450 Enzyme InhibitorsDisease Models, AnimalDogsEther-A-Go-Go Potassium Channels--antagonists & inhibitorsHEK293 CellsHeart--drug effectsHistamine H3 Antagonists--adverse effectsHumansMaleNeuralgia--drug therapyOsteoarthritis--drug therapyOsteoarthritis, Knee--drug therapyPyridazines--adverse effectsRatsRats, Sprague-DawleyReceptors, Histamine H3--metabolismSubstrate Specificity